Catalogue Number: CV-1010-2-RPE
Manufacturer: | rPeptide |
Physical state: | Lyophilized |
Type: | Other Inhibitors |
Shipping Condition: | RT |
Unit(s): | 25 mg |
Description: RVX-208 is a potent BET bromodomain antagonist with IC50 of 0.510 µM for BD2, with approximately 170-fold selectivity over BD1. Increases apolipoprotein A-1 and HDL cholesterol in vitro and in vivo Reduces atherosclerosis.