dBET57

Catalogue Number: S0137-SEL

Manufacturer:Selleck Chemicals
Molecular Formula:C34H31ClN8O5S
Type:Biochemicals
Shipping Condition:Blue Ice
Unit(s): 25 mg, 5 mg

Additional Text

Short Description

dBET57 is a novel, potent and selective degrader of BRD4BD1 based on the PROTAC technology with DC50/5h of 500 nM. dBET57 is inactive on BRD4BD2.

Smile String

CC1=C(SC2=C1C(=NC(C3=NN=C(N32)C)CC(=O)NCCNC4=CC=CC5=C4C(=O)N(C5=O)C6CCC(=O)NC6=O)C7=CC=C(C=C7)Cl)C

Storage Note

3 years -20°C powder