Catalogue Number: S0717-SEL
Manufacturer: | Selleck Chemicals |
Type: | Biochemicals |
Shipping Condition: | Blue Ice |
Unit(s): | 5 mg |
Description: Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR)and α3β4 nAChRwith EC50 of 2.3 µM and 55 µM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRswith EC50 of 18 µM. Varenicline is a prescription medication used for smoking cessation.