Varenicline (CP 526555) dihydrochloride

Catalogue Number: S0717-SEL

Manufacturer:Selleck Chemicals
Type:Biochemicals
Shipping Condition:Blue Ice
Unit(s): 5 mg

Description

Description: Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 µM and 55 µM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 µM. Varenicline is a prescription medication used for smoking cessation.