Catalogue Number: S1216-SEL
Manufacturer: | Selleck Chemicals |
Shelf Life: | 24 months |
Molecular Formula: | C16H17N3O4S |
Type: | Other Inhibitors |
Shipping Condition: | Blue Ice |
Unit(s): | 5 mg, 1 g |
FOR RESEARCH USE ONLY
PFI-1 (PF-6405761) is a highly selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 µM and for BRD2 with IC50 of 98 nM in a cell-free assay.
CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O
2 years -80 in solvent