PFI-1 (PF-6405761)

Catalogue Number: S1216-SEL

Manufacturer:Selleck Chemicals
Shelf Life:24 months
Molecular Formula:C16H17N3O4S
Type:Other Inhibitors
Shipping Condition:Blue Ice
Unit(s): 5 mg, 1 g

Additional Text

Caution

FOR RESEARCH USE ONLY

Short Description

PFI-1 (PF-6405761) is a highly selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 µM and for BRD2 with IC50 of 98 nM in a cell-free assay.

Smile String

CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O

Storage Note

2 years -80 in solvent