Catalogue Number: S1421-SEL
Manufacturer: | Selleck Chemicals |
Physical state: | Lyophilized |
Type: | Other Inhibitors |
Alias: | Staurosporine |
Shipping Condition: | Blue Ice |
Unit(s): | 2 mg, 5 mg, 25 mg, 1 g, 10 mM/1 ml |
Description: Staurosporine (STS) is a potent PKCinhibitor for PKCα, PKCγ and PKCη with IC50of 2 nM, 5 nM and 4 nM, less potent to PKCδ (20 nM), PKCε (73 nM) and little active to PKCζ (1086 nM) in cell-free assays. Also shows inhibitory activities on other kinases, such as PKA, PKG, S6K, CaMKII, etc. Phase 3.
FOR RESEARCH USE ONLY