Catalogue Number: S8532-SEL
Manufacturer: | Selleck Chemicals |
Type: | Biochemicals |
Shipping Condition: | Blue Ice |
Unit(s): | 1 mg, 5 mg, 10 mM/1 ml, 1 g, 100 mg, 25 mg |
Description: ARV-771 is a potent pan-(bromodomain and extra-terminal)BETdegrader, a novel BET-PROTAC(proteolysis-targeting chimera) with Kd of 34 nM, 4.7 nM, 8.3 nM, 7.6 nM, 9.6 nM, and 7.6 nM for BRD2(1), BRD2(2), BRD3(1), BRD3(2), BRD4(1), and BRD4(2), respectively.